KinomeScan

KINOMEscan™ - Explore Our Panel

Expand each group to select individual kinases. Those marked with an asterisk (*) do not appear on tree. Request a Quote
 

All Available Kinases

Click to ExpandAGC

Select All 38
AKT1 AKT2 AKT3 CIT
DMPK DMPK2 GRK1 GRK4
GRK7 LATS1
LATS2 MAST1 MRCKA MRCKB
NDR1 NDR2 PDPK1 PKAC-alpha
PKAC-beta PKN1 PKN2 PRKCD
PRKCE PRKCH PRKCQ PRKG1
PRKG2 PRKX ROCK1 ROCK2
RPS6KA1(Kin.Dom.1-N-terminal)
RPS6KA2(Kin.Dom.1-N-terminal)
RPS6KA3(Kin.Dom.1-N-terminal)
RPS6KA4(Kin.Dom.1-N-terminal)
RPS6KA5(Kin.Dom.1-N-terminal)
RPS6KA6(Kin.Dom.1-N-terminal)
YANK2 YANK3

Click to ExpandCAMK

Select All 58
AMPK-alpha1 AMPK-alpha2 ARK5
BRSK1 BRSK2 CAMK1 CAMK1D CAMK1G
CAMK2A CAMK2B CAMK2D CAMK2G CAMK4
CHEK1 CHEK2 DAPK1 DAPK2 DAPK3
DCAMKL1 DCAMKL2 DCAMKL3 DRAK1 DRAK2
HUNK LKB1 MAPKAPK2 MAPKAPK5 MARK1
MARK2 MARK3 MARK4 MELK MKNK1
MKNK2 MLCK MYLK MYLK2 NIM1
PHKG1 PHKG2
PIM1 PIM2 PIM3 PRKD1 PRKD2
PRKD3 QSK RPS6KA1(Kin.Dom.2-C-terminal)
RPS6KA2(Kin.Dom.2-C-terminal)
RPS6KA4(Kin.Dom.2-C-terminal)
RPS6KA5(Kin.Dom.2-C-terminal)
RPS6KA6(Kin.Dom.2-C-terminal) SIK
SIK2 SgK085 SNARK STK33 TSSK1B

Click to ExpandCK1

Select All 6
CSNK1A1L CSNK1D CSNK1E CSNK1G1 CSNK1G2
CSNK1G3

Click to ExpandCMGC

Select All 50
CDC2L1 CDC2L2* CDK11 CDK2 CDK3
CDK5 CDK7 CDK8 CDK9 CDKL2
CDKL3 CDKL5 CLK1 CLK2 CLK3
CLK4 DYRK1A DYRK1B DYRK2 ERK1
ERK2 ERK3 ERK4 ERK5 ERK8
GSK3A GSK3B HIPK1 HIPK2
HIPK3 HIPK4 ICK JNK1 JNK2
JNK3 MAK NLK p38-alpha
p38-beta p38-delta p38-gamma PCTK1
PCTK2 PCTK3 PFTAIRE2 PFTK1 PRP4
SRPK1 SRPK2 SRPK3

Click to ExpandSTE

Select All 40
ASK1 ASK2 HPK1 LOK MAP3K1
MAP3K15 MAP3K2 MAP3K3 MAP3K4 MAP4K2
MAP4K3 MAP4K4 MAP4K5 MEK1 MEK2
MEK3 MEK4 MEK6 MINK MST1
MST2 MST3 MST4 MYO3A MYO3B
OSR1 PAK1 PAK2 PAK3 PAK4
PAK6 PAK7 SLK STK39 TAO1
TAOK1 TAOK3 TNIK YSK1 YSK4

Click to ExpandTK

Select All 83
ABL1 ABL2 ALK AXL BLK
BMX BRK BTK CSF1R CSK
CTK DDR1 DDR2 EGFR EPHA1
EPHA2 EPHA3 EPHA4 EPHA5 EPHA6
EPHA7 EPHA8 EPHB1 EPHB2 EPHB3
EPHB4 EPHB6 ERBB2 ERBB3 ERBB4
FAK FER FES FGFR1 FGFR2
FGFR3 FGFR4 FGR FLT1 FLT3
FLT4 FRK FYN HCK IGF1R
INSR INSRR ITK
JAK1(JH2domain-pseudokinase)
JAK1(JH1domain-catalytic)
JAK2(JH1domain-catalytic)
JAK3(JH1domain-catalytic)
KIT LCK LTK LYN MERTK
MET MST1R MUSK PDGFRA PDGFRB
PYK2 RET ROS1 SRC SRMS
SYK TEC TIE1 TIE2 TNK1
TNK2 TRKA TRKB TRKC TXK
TYK2(JH1domain-pseudokinase)
TYK2(JH1domain-catalytic)
TYRO3 VEGFR2 YES ZAP70

Click to ExpandTKL

Select All 29
ACVR1 ACVR1B ACVR2A ACVR2B ACVRL1
ANKK1 BMPR1A BMPR1B BMPR2 BRAF
DLK IRAK1 IRAK3 LIMK1 LIMK2
LZK MLK1 MLK2 MLK3 RAF1
RIPK1 RIPK2 RIPK4 TAK1 TESK1
TGFBR1 TGFBR2 TNNI3K ZAK

Click to ExpandATYPICAL*

Select All 5
ADCK3 ADCK4
RIOK1 RIOK2 RIOK3

Click to ExpandMUTANT*

Select All 36
ABL1(E255K) ABL1(F317I) ABL1(F317L)
ABL1(H396P) ABL1(M351T) ABL1(Q252H)
ABL1(T315I) ABL1(Y253F)
EGFR(E746-A750del) EGFR(G719C)
EGFR(L747-E749del,A750P) EGFR(G719S)
EGFR(L747-S752del,P753S) EGFR(L858R)
EGFR(L858R,T790M)
EGFR(L747-T751del,Sins)
EGFR(L861Q) EGFR(S752-I759del)
FGFR3(G697C) FLT3(D835H) FLT3(D835Y)
FLT3(ITD) FLT3(K663Q) FLT3(N841I)
KIT(D816V) KIT(L576P) KIT(V559D)
KIT(V559D,T670I) KIT(V559D,V654A) MET(M1250T)
MET(Y1235D) PIK3CA(E545K) RET(M918T)
RET(V804L) RET(V804M) BRAF(V600E)

Click to ExpandLIPID*

Select All 16
PIK3C2B PIK3C2G PIK3CA
PIK3CA(C420R) PIK3CA(E542K) PIK3CA(E545A)
PIK3CA(H1047L) PIK3CA(H1047Y) PIK3CA(M1043I)
PIK3CA(Q546K) PIK3CB PIK3CD
PIK3CG PIK4CB PIP5K1A
PIP5K2B

Click to ExpandOTHER

Select All 41
AAK1 AURKA AURKB AURKC BIKE
CAMKK1 CAMKK2 CSNK2A1 CSNK2A2 ERN1
GAK GCN2(Kin.Dom.2,S808G) IKK-alpha
IKK-beta IKK-epsilon NEK1 NEK2
NEK5 NEK6 NEK7 NEK9 PKMYT1
PLK1 PLK2 PLK3 PLK4 PRKR
SBK1 SGK110 STK16 STK35 STK36
TBK1 TLK1 TLK2 TTK ULK1
ULK2 ULK3 WEE1 WEE2

Human Kinome image created and provided by Cell Signaling Technology, Inc. Cell Signaling


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